Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50019795
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50617567(CHEMBL5395794)
Affinity DataKd:  120nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) at 100 uM by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623073(CHEMBL5410133)
Affinity DataKd:  160nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) at 100 uM by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataKd:  100nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) at 100 uM by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50617569(CHEMBL5418436)
Affinity DataIC50: 25nMAssay Description:Inhibition of N-terminal StrepII-SUMO or SUMO-AviTag/Cterminal 6xHis tagged ENL (unknown origin) (1 to 148 residues) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623091(CHEMBL5437942)
Affinity DataIC50: 40nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50617567(CHEMBL5395794)
Affinity DataIC50: 50nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataIC50: 120nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623072(CHEMBL5434752)
Affinity DataIC50: 130nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623080(CHEMBL5430048)
Affinity DataIC50: 130nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623082(CHEMBL5434666)
Affinity DataIC50: 150nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623081(CHEMBL5423084)
Affinity DataIC50: 170nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623074(CHEMBL5437279)
Affinity DataIC50: 180nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623073(CHEMBL5410133)
Affinity DataIC50: 190nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623075(CHEMBL5423179)
Affinity DataIC50: 260nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataIC50: 260nMAssay Description:Inhibition of wild type human ENL YEATS expressed in Escherichia coli Rosetta cells by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623083(CHEMBL5403490)
Affinity DataIC50: 280nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623078(CHEMBL5395504)
Affinity DataIC50: 350nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623089(CHEMBL5394853)
Affinity DataIC50: 360nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623079(CHEMBL5396023)
Affinity DataIC50: 380nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623077(CHEMBL5435284)
Affinity DataIC50: 390nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623071(CHEMBL5440223)
Affinity DataIC50: 490nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623092(CHEMBL5417885)
Affinity DataIC50: 560nMAssay Description:Inhibition of ENT YEATS domain (unknown origin) using photo-H3K9cr as substrate by competitive photo-cross-linking methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623085(CHEMBL5396726)
Affinity DataIC50: 630nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623090(CHEMBL5395927)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623086(CHEMBL5428403)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623084(CHEMBL5420102)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623076(CHEMBL5411970)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623087(CHEMBL5411434)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
Sanders Tri-Institutional Therapeutics

Curated by ChEMBL
LigandPNGBDBM50623088(CHEMBL5422746)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed