Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50019626
LigandPNGBDBM50621141(CHEMBL5427257)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of His-tagged PD-1 (unknown origin)/hFc-tagged PD-L1 (unknown origin) protein-protein interaction incubated for 15 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621143(CHEMBL5423533)
Affinity DataIC50: 1nMAssay Description:Inhibition of His-tagged PD-1 (unknown origin)/hFc-tagged PD-L1 (unknown origin) protein-protein interaction incubated for 15 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50239948(US9850225, Example 1166 | CHEMBL4071326)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of C-terminal 3S-IG-tagged recombinant human PD-1 (25 to 167 residues)/C-terminal 6xHis-tagged recombinant human PD-L1 (18 to 239 residues...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM363065(US9850225, Example 1002 | (R)-2-(2-(3-cyanobenzylo...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of C-terminal 3S-IG-tagged recombinant human PD-1 (25 to 167 residues)/C-terminal 6xHis-tagged recombinant human PD-L1 (18 to 239 residues...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621158(CHEMBL5419797)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621174(CHEMBL5412235)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621155(CHEMBL5432909)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50239942(US9872852, Example 37 | CHEMBL4081869)
Affinity DataIC50: 6nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM366037(N-(2-{[(4-{[3-(2,3-dihydro-1,4- benzodioxin-6-yl)-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621161(CHEMBL5436822)
Affinity DataIC50: 6nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM365801(1-({3-methyl-4-[(2-methyl-3- phenylphenyl)methoxy]...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621152(CHEMBL5425865)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621164(CHEMBL5436514)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50542963(CHEMBL4638650)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621154(CHEMBL5424869)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621157(CHEMBL5414835)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621153(CHEMBL5430973)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621166(CHEMBL5416482)
Affinity DataIC50: 10nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621142(CHEMBL5411833)
Affinity DataIC50: 10nMAssay Description:Inhibition of His-tagged PD-1 (unknown origin)/hFc-tagged PD-L1 (unknown origin) protein-protein interaction incubated for 15 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM363328(N-(2-((5-chloro-2-((3-cyanobenzyl)oxy)-4-((3-(2,3-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621170(CHEMBL5424916)
Affinity DataIC50: 12nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621172(CHEMBL5412039)
Affinity DataIC50: 12nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621160(CHEMBL5400124)
Affinity DataIC50: 16nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621169(CHEMBL5426426)
Affinity DataIC50: 16nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50239947(US9872852, Example 202 | CHEMBL4089730 | US2023030...)
Affinity DataIC50: 18nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621167(CHEMBL5439310)
Affinity DataIC50: 19nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621163(CHEMBL5410844)
Affinity DataIC50: 29nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621165(CHEMBL5396887)
Affinity DataIC50: 30nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621156(CHEMBL5398595)
Affinity DataIC50: 46nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621162(CHEMBL5408386)
Affinity DataIC50: 50nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621159(CHEMBL5408730)
Affinity DataIC50: 50nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50239947(US9872852, Example 202 | CHEMBL4089730 | US2023030...)
Affinity DataIC50: 101nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM366034(N-(2-{[(4-{[3- (3-ethoxyphenyl)-2- methylphenyl]me...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM366035(N-(2-{[(4-{[3-(2H-1,3- benzodioxol-5-yl)-2- methyl...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM365798(1-({3-fluoro-4-[(2-methyl-3- phenylphenyl)methoxy]...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM365965(N-{2-[({6-[(2-methyl-3- phenylphenyl)methoxy]pyrid...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM363425(US9850225, Example 1335 | N-(2-((2-methoxy-4-((2-m...)
Affinity DataIC50: 110nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50239943(US9872852, Example 8 | CHEMBL4099869)
Affinity DataIC50: 146nMAssay Description:Inhibition of Ig-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) protein-protein interaction preincubated with PD-L1 for 15 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50091334(CHEMBL3582252)
Affinity DataIC50: 202nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621147(CHEMBL5429159)
Affinity DataIC50: 207nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621168(CHEMBL5398056)
Affinity DataIC50: 589nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621171(CHEMBL5422336)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621146(CHEMBL5418648)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621173(CHEMBL5440112)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621150(CHEMBL5424402)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621148(CHEMBL5436818)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621149(CHEMBL5423262)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621151(CHEMBL5434250)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621144(CHEMBL5414313)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50621145(CHEMBL5427994)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PD-1 binding to human PD-L1 by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
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