Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50021475
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641046(CHEMBL5568763)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641032(CHEMBL5575395)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641055(CHEMBL5595017)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641050(CHEMBL5542251)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641054(CHEMBL5594953)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641031(CHEMBL5574827)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641052(CHEMBL5570575)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641034(CHEMBL5569106)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641053(CHEMBL5570942)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641049(CHEMBL5571583)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641039(CHEMBL5591422)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641042(CHEMBL5570541)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641051(CHEMBL5593626)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641051(CHEMBL5593626)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641044(CHEMBL5549815)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641039(CHEMBL5591422)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641055(CHEMBL5595017)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641050(CHEMBL5542251)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641033(CHEMBL5572790)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641052(CHEMBL5570575)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641048(CHEMBL5572703)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641045(CHEMBL5570657)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641043(CHEMBL5569619)
Affinity DataKi:  4.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641032(CHEMBL5575395)
Affinity DataKi:  5.10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641054(CHEMBL5594953)
Affinity DataKi:  5.70nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641045(CHEMBL5570657)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641035(CHEMBL5572310)
Affinity DataKi:  6.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641049(CHEMBL5571583)
Affinity DataKi:  7.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641037(CHEMBL5569227)
Affinity DataKi:  7.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641046(CHEMBL5568763)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641036(CHEMBL5594507)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641040(CHEMBL5574967)
Affinity DataKi:  8.60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641048(CHEMBL5572703)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641043(CHEMBL5569619)
Affinity DataKi:  9.40nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641044(CHEMBL5549815)
Affinity DataKi:  9.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50615426(CHEMBL5274078)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641033(CHEMBL5572790)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641038(CHEMBL5570330)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641041(CHEMBL5563699)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Human)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641041(CHEMBL5563699)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641035(CHEMBL5572310)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641040(CHEMBL5574967)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641034(CHEMBL5569106)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641042(CHEMBL5570541)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641053(CHEMBL5570942)
Affinity DataKi:  26nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641047(CHEMBL5571001)
Affinity DataKi:  29nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641031(CHEMBL5574827)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641036(CHEMBL5594507)
Affinity DataKi:  37nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50615426(CHEMBL5274078)
Affinity DataKi:  39nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistamine H3 receptor(Rat)
Gedeon Richter Plc.

Curated by ChEMBL
LigandPNGBDBM50641037(CHEMBL5569227)
Affinity DataKi:  55nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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