Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50020597
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631710(CHEMBL5426932)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631712(CHEMBL5399482)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631708(CHEMBL5409299)
Affinity DataIC50: 3.17E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631713(CHEMBL5437506)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631709(CHEMBL5402786)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631714(CHEMBL5394140)
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631711(CHEMBL5405630)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50242284(scutellarin | CHEMBL487805)
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631707(CHEMBL5403462)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631715(CHEMBL5420251)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631716(CHEMBL5417022)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631717(CHEMBL5400953)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50631718(CHEMBL5401400)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant P-gp ATPase activity in isolated membranes incubated in presence of verapamil by firefly luciferase based luminescenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed