Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50019607
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal HA-tagged recombinant wild-type human MLK3 overexpressed in HEK293A cells preincubated for 10 mins followed by [gamma-32P]AT...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of N-terminal GST-tagged recombinant MLK3 (unknown origin) expressed in insect cells incubated for 15 mins in presence of [gamma-32P]ATP b...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of MLK3 (unknown origin) by cell-free radiolabeled ATP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of human MLK3 by ATP-competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Chungnam National University
Curated by ChEMBL
Chungnam National University
Curated by ChEMBL
Affinity DataIC50: 5.92E+3nMAssay Description:Inhibition of MLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
