Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50020069
Target5-hydroxytryptamine receptor 2B(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625921(CHEMBL5409958)
Affinity DataKi:  500nMAssay Description:Inhibition of human 5-HT2B receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625925(CHEMBL5396440)
Affinity DataKi:  550nMAssay Description:Inhibition of human 5-HT2B receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625928(CHEMBL5412183)
Affinity DataKi:  620nMAssay Description:Inhibition of human 5-HT2B receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625924(CHEMBL5418175)
Affinity DataKi:  710nMAssay Description:Inhibition of human 5-HT2B receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625926(CHEMBL5411964)
Affinity DataKi:  830nMAssay Description:Inhibition of human 5-HT2B receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625921(CHEMBL5409958)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human 5-HT6 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625929(CHEMBL5400817)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human 5-HT2B receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625921(CHEMBL5409958)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human KOR assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625924(CHEMBL5418175)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of human sigma 2 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetKappa-type opioid receptor(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625923(CHEMBL5397467)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human KOR assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625926(CHEMBL5411964)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of human sigma 1 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625921(CHEMBL5409958)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human alpha 2C adrenergic receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625925(CHEMBL5396440)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of human 5-HT1D receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625927(CHEMBL5435643)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of human 5-HT1D receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625921(CHEMBL5409958)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of human sigma 1 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625925(CHEMBL5396440)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human sigma 1 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625925(CHEMBL5396440)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human sigma 2 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625922(CHEMBL5422761)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human sigma 2 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625922(CHEMBL5422761)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of human sigma 1 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625923(CHEMBL5397467)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of human sigma 2 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50625923(CHEMBL5397467)
Affinity DataKi:  6.50E+3nMAssay Description:Inhibition of human sigma 1 receptor assessed as inhibition constant by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed