Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50020999
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50519651(CHEMBL4534082)
Affinity DataKd:  400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50602054(CHEMBL5209456)
Affinity DataKd:  15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataKd:  100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50602054(CHEMBL5209456)
Affinity DataKd: >5.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635880(CHEMBL5568050)
Affinity DataKd:  209nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM26474(GW-786034 | JMC514632 Compound 13 | 5-({4-[(2,3-di...)
Affinity DataKd:  260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50323777(N-(4-Methyl-3-(1-methyl-7-(6-methylpyridin-3-ylami...)
Affinity DataKd:  56nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM31084(1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-...)
Affinity DataKd:  1.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635880(CHEMBL5568050)
Affinity DataKd:  199nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635875(CHEMBL5518057)
Affinity DataKd:  13nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635879(CHEMBL5517778)
Affinity DataKd:  8.70nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50322535(3-[2-(Imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-meth...)
Affinity DataKd:  37nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50519641(CHEMBL4439426)
Affinity DataKd:  218nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50602055(CHEMBL5182551)
Affinity DataKd:  78nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetRegulator of chromosome condensation(Homo sapiens)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM185674(Rebastinib | 4-[4-[(5-tert-butyl-2-quinolin-6-ylpy...)
Affinity DataEC50:  19nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635882(CHEMBL5565328)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50442165(CHEMBL2441341)
Affinity DataIC50: 3.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50513014(CHEMBL4442060)
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635875(CHEMBL5518057)
Affinity DataIC50: 5.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM185674(Rebastinib | 4-[4-[(5-tert-butyl-2-quinolin-6-ylpy...)
Affinity DataIC50: 6.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataIC50: 6.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50442167(CHEMBL2441339)
Affinity DataIC50: 9.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50263058(CHEMBL4090723)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50065454(CHEMBL3348846 | CHEBI:63453)
Affinity DataIC50: 12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50113499(CHEMBL3604619)
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50442165(CHEMBL2441341)
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM185674(Rebastinib | 4-[4-[(5-tert-butyl-2-quinolin-6-ylpy...)
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50323777(N-(4-Methyl-3-(1-methyl-7-(6-methylpyridin-3-ylami...)
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50323777(N-(4-Methyl-3-(1-methyl-7-(6-methylpyridin-3-ylami...)
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase A(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50355496(CHEMBL1908397)
Affinity DataIC50: 48nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50442167(CHEMBL2441339)
Affinity DataIC50: 69nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635877(CHEMBL5537068)
Affinity DataIC50: 90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635877(CHEMBL5537068)
Affinity DataIC50: 90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM31084(1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-(2-fluoro-...)
Affinity DataIC50: 95nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM423400(US10501473, Example 39)
Affinity DataIC50: 110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635881(CHEMBL5556669)
Affinity DataIC50: 160nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50263059(CHEMBL4105556)
Affinity DataIC50: 170nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635876(CHEMBL5567128)
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 2(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50065454(CHEMBL3348846 | CHEBI:63453)
Affinity DataIC50: 259nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase A(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50263059(CHEMBL4105556)
Affinity DataIC50: 293nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635874(CHEMBL365607)
Affinity DataIC50: 320nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635878(CHEMBL5567010)
Affinity DataIC50: 366nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635878(CHEMBL5567010)
Affinity DataIC50: 366nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetAurora kinase A(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50635881(CHEMBL5556669)
Affinity DataIC50: 430nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataIC50: 618nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataIC50: 618nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50322535(3-[2-(Imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-meth...)
Affinity DataIC50: 640nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50263057(CHEMBL381230)
Affinity DataIC50: 910nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM50519641(CHEMBL4439426)
Affinity DataIC50: 1.03E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Lanzhou University Second Hospital

Curated by ChEMBL
LigandPNGBDBM36371(CID2828334 | 5-(1H-indol-3-ylmethyl)-3-methyl-2-th...)
Affinity DataIC50: 1.98E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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