Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019769
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622924(CHEMBL5402846)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate preincubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622925(CHEMBL5401123)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate preincubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622923(CHEMBL5414105)
Affinity DataIC50: 2.05E+4nMAssay Description:Inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate preincubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622922(CHEMBL5426441)
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate preincubated for ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622921(CHEMBL5417828)
Affinity DataIC50: 5.46E+4nMAssay Description:Inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate preincubated for ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622924(CHEMBL5402846)
Affinity DataKi:  200nMAssay Description:Competitive inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622925(CHEMBL5401123)
Affinity DataKi:  800nMAssay Description:Competitive inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTrypanothione reductase(Leishmania infantum)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50622923(CHEMBL5414105)
Affinity DataKi:  5.50E+3nMAssay Description:Competitive inhibition of Leishmania infantum Trypanothione reductase expressed in Escherichia coli BL21 (DE3) using trypanothione as substrate prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed