Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50020059
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625880(CHEMBL5396548)
Affinity DataEC50:  2.11E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625890(CHEMBL5418881)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625889(CHEMBL5419687)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625888(CHEMBL5415308)
Affinity DataEC50:  1.04E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625887(CHEMBL5395068)
Affinity DataEC50:  1.56E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625886(CHEMBL5428833)
Affinity DataEC50:  481nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625885(CHEMBL5419801)
Affinity DataEC50:  885nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625884(CHEMBL5412687)
Affinity DataEC50:  9.00E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625883(CHEMBL5432025)
Affinity DataEC50:  1.07E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625882(CHEMBL5440040)
Affinity DataEC50:  6.50E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625881(CHEMBL5414380)
Affinity DataEC50:  1.87E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625869(CHEMBL5432101)
Affinity DataEC50:  675nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625879(CHEMBL5424688)
Affinity DataEC50:  3.69E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625878(CHEMBL5406419)
Affinity DataEC50:  2.60E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625877(CHEMBL5409056)
Affinity DataEC50: >4.88E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625876(CHEMBL5422473)
Affinity DataEC50: >4.88E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625875(CHEMBL5415347)
Affinity DataEC50: >4.88E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625874(CHEMBL5423474)
Affinity DataEC50: >4.88E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625873(CHEMBL5430756)
Affinity DataEC50:  2.24E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625872(CHEMBL5440855)
Affinity DataEC50:  3.48E+3nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625871(CHEMBL5407879)
Affinity DataEC50:  1.24E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMucolipin-2(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50625870(CHEMBL5428524)
Affinity DataEC50: >4.88E+4nMAssay Description:Agonist activity at human TRPML1 expressed in HEK293 cells incubated for 1 hr by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed