Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50021519
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641492(CHEMBL5569161)
Affinity DataIC50: 111nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641496(CHEMBL5568622)
Affinity DataIC50: 135nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641476(CHEMBL5567043)
Affinity DataIC50: 136nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641488(CHEMBL5563043)
Affinity DataIC50: 155nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641501(CHEMBL5590984)
Affinity DataIC50: 164nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 186nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641486(CHEMBL5569094)
Affinity DataIC50: 196nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641475(CHEMBL5555360)
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641463(CHEMBL5565769)
Affinity DataIC50: 212nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641503(CHEMBL5565943)
Affinity DataIC50: 214nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641474(CHEMBL5575877)
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641473(CHEMBL5593403)
Affinity DataIC50: 295nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641465(CHEMBL5593664)
Affinity DataIC50: 332nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641494(CHEMBL5563792)
Affinity DataIC50: 443nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641498(CHEMBL5570562)
Affinity DataIC50: 452nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641502(CHEMBL5594723)
Affinity DataIC50: 461nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641467(CHEMBL5573730)
Affinity DataIC50: 505nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641485(CHEMBL5571572)
Affinity DataIC50: 544nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641495(CHEMBL5573769)
Affinity DataIC50: 597nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641487(CHEMBL5571059)
Affinity DataIC50: 625nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641470(CHEMBL5571115)
Affinity DataIC50: 655nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641489(CHEMBL5574997)
Affinity DataIC50: 716nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641472(CHEMBL5563225)
Affinity DataIC50: 792nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641466(CHEMBL5589667)
Affinity DataIC50: 806nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641456(CHEMBL5574098)
Affinity DataIC50: 831nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641457(CHEMBL5594380)
Affinity DataIC50: 999nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641469(CHEMBL5563558)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641497(CHEMBL5574051)
Affinity DataIC50: 1.06E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641483(CHEMBL5572979)
Affinity DataIC50: 1.08E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641458(CHEMBL5572389)
Affinity DataIC50: 1.10E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641460(CHEMBL5584051)
Affinity DataIC50: 1.13E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641468(CHEMBL5569474)
Affinity DataIC50: 1.14E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641493(CHEMBL5565870)
Affinity DataIC50: 1.15E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641481(CHEMBL5571579)
Affinity DataIC50: 1.23E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641491(CHEMBL5572527)
Affinity DataIC50: 1.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641462(CHEMBL5572462)
Affinity DataIC50: 1.32E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641464(CHEMBL5574403)
Affinity DataIC50: 1.42E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641499(CHEMBL5573540)
Affinity DataIC50: 1.54E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641471(CHEMBL5566095)
Affinity DataIC50: 1.58E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641490(CHEMBL5564844)
Affinity DataIC50: 1.59E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641461(CHEMBL5571658)
Affinity DataIC50: 1.63E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641484(CHEMBL5564208)
Affinity DataIC50: 1.64E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641455(CHEMBL5572524)
Affinity DataIC50: 1.76E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641480(CHEMBL5574257)
Affinity DataIC50: 2.58E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641500(CHEMBL5590394)
Affinity DataIC50: 2.61E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641477(CHEMBL5574975)
Affinity DataIC50: 3.14E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641478(CHEMBL5565106)
Affinity DataIC50: 3.38E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641496(CHEMBL5568622)
Affinity DataIC50: 3.50E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641459(CHEMBL5574056)
Affinity DataIC50: 4.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641479(CHEMBL5569875)
Affinity DataIC50: 5.03E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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