Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50020492
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630453(CHEMBL5403846)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630463(CHEMBL5418976)
Affinity DataKd:  340nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630462(CHEMBL5431869)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630461(CHEMBL5432199)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630460(CHEMBL5432238)
Affinity DataKd:  6.90E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630459(CHEMBL5415641)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630458(CHEMBL5409882)
Affinity DataKd:  6.90E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630457(CHEMBL5434964)
Affinity DataKd:  6.90E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630456(CHEMBL5433508)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630455(CHEMBL5424624)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630454(CHEMBL5398410)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50293523(N-(1H-benzo[d][1,2,3]triazol-6-yl)-2-(6-methylpyri...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50293516(2-(6-methylpyridin-2-yl)-N-(pyridin-4-yl)quinazoli...)
Affinity DataKd:  10nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50293521(N-(1-methyl-1H-indazol-5-yl)-2-(6-methylpyridin-2-...)
Affinity DataKd:  5.50E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630452(CHEMBL5400594)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630451(CHEMBL5424398)
Affinity DataKd:  8.90E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630450(CHEMBL5424567)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630449(CHEMBL5432948)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630448(CHEMBL5425571)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630447(CHEMBL5426158)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630446(CHEMBL5406226)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50630445(CHEMBL5429572)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetTGF-beta receptor type-1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50293522(N-(2-(6-methylpyridin-2-yl)quinazolin-4-yl)benzo[d...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to wild type human partial length TGFBR1 (D179 to M503 residues) expressed in bacterial expression system by KINOMEscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed