Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50020841
TargetTyrosine-protein kinase JAK2(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM99537(CHEMBL2062804 | US8501936, 35)
Affinity DataIC50: 6nMAssay Description:Inhibition of JAK2 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM99537(CHEMBL2062804 | US8501936, 35)
Affinity DataIC50: 12nMAssay Description:Inhibition of JAK1 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634010(CHEMBL5419546)
Affinity DataIC50: 74nMAssay Description:Inhibition of JAK2 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM99537(CHEMBL2062804 | US8501936, 35)
Affinity DataIC50: 86nMAssay Description:Inhibition of JAK3 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634011(CHEMBL5419117)
Affinity DataIC50: 90nMAssay Description:Inhibition of JAK2 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634009(CHEMBL5435274)
Affinity DataIC50: 326nMAssay Description:Inhibition of JAK2 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634013(CHEMBL5402252)
Affinity DataIC50: 544nMAssay Description:Inhibition of JAK2 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634012(CHEMBL5436068)
Affinity DataIC50: 705nMAssay Description:Inhibition of JAK2 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTubulin beta chain(Pig)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634010(CHEMBL5419546)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured for 30 mins in presence of GTP by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTubulin beta chain(Pig)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634012(CHEMBL5436068)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured for 30 mins in presence of GTP by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTubulin beta chain(Pig)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634009(CHEMBL5435274)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured for 30 mins in presence of GTP by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTubulin beta chain(Pig)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50014846(7alphaH-colchicine | (S)-N-(5,6,7,9-tetrahydro-1,2...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured for 30 mins in presence of GTP by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTubulin beta chain(Pig)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634011(CHEMBL5419117)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization measured for 30 mins in presence of GTP by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634010(CHEMBL5419546)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of JAK3 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTubulin beta chain(Pig)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634013(CHEMBL5402252)
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization measured for 30 mins in presence of GTP by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK1(Human)
Wuyi University

Curated by ChEMBL
LigandPNGBDBM50634010(CHEMBL5419546)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of JAK1 (unknown origin) using Poly-(Glu,Tyr 4:1) peptide as substrate in presence of ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed