Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50019598
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620854(CHEMBL5421022)
Affinity DataIC50: 25nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620851(CHEMBL5421003)
Affinity DataIC50: 70nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620857(CHEMBL5400244)
Affinity DataIC50: 90nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620858(CHEMBL5393802)
Affinity DataIC50: 150nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620855(CHEMBL5411351)
Affinity DataIC50: 160nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620852(CHEMBL5434711)
Affinity DataIC50: 170nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620865(CHEMBL5419063)
Affinity DataIC50: 310nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620859(CHEMBL5409298)
Affinity DataIC50: 390nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620862(CHEMBL5428824)
Affinity DataIC50: 400nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM40402(cid_1185399 | 2-furancarboxylic acid [3-(2-methoxy...)
Affinity DataIC50: 440nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620856(CHEMBL5404501)
Affinity DataIC50: 490nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620861(CHEMBL5400240)
Affinity DataIC50: 800nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620853(CHEMBL5434719)
Affinity DataIC50: 800nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620860(CHEMBL5405353)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM40404(acetic acid [6-ethyl-2-methyl-3-(1-methyl-2-benzim...)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM37759([3-(2-methoxyphenyl)-2-methyl-4-oxidanylidene-chro...)
Affinity DataIC50: 1.90E+3nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620866(CHEMBL1424418)
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620863(CHEMBL5431353)
Affinity DataIC50: 2.19E+4nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetfMet-Leu-Phe receptor(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50620864(CHEMBL5437205)
Affinity DataIC50: 2.89E+4nMAssay Description:Antagonist activity against human FPR1 expressed in human HL-60 cells assessed as inhibition of fMLF-induced calcium mobilization preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed