Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50020451
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 9.60E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 62nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 3.20E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 650nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 2.90E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.20E+4nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 620nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 68nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 4.70E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
