Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50020316
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628765(CHEMBL5415486)
Affinity DataIC50: 0.410nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628766(CHEMBL5433360)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628764(CHEMBL5418103)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628768(CHEMBL5398070)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628769(CHEMBL5428323)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628771(CHEMBL5407739)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628766(CHEMBL5433360)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628765(CHEMBL5415486)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628770(CHEMBL5413614)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628764(CHEMBL5418103)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628771(CHEMBL5407739)
Affinity DataIC50: 69nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628767(CHEMBL5418493)
Affinity DataIC50: 81nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628769(CHEMBL5428323)
Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628768(CHEMBL5398070)
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628770(CHEMBL5413614)
Affinity DataIC50: 430nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628772(CHEMBL5401618)
Affinity DataIC50: 710nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628767(CHEMBL5418493)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetEnteropeptidase(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50628772(CHEMBL5401618)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human recombinant enteropeptidase using 5FAM-Abu-Gly-Asp-Asp-Asp-Lys-Ile-Val-Gly-Gly-Lys(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed