Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50020306
Affinity DataIC50: 7.40nMAssay Description:Inhibition of EGFR-D770-N771insNPG mutant (unknown origin) phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of wildtype EGFR (unknown origin) phosphorylationMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity to EGFR-A763-Y764insFQEA mutant (unknown origin) assessed as inhibition constant in presence of ATPMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 6.40nMAssay Description:Binding affinity to EGFR L858R mutant (unknown origin) assessed as inhibition constant in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to human EGFR L858R/T790M mutant (696 to 1022 residues) expressed in insect cells assessed as inhibition constant in presence of ATP...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to wildtype EGFR (unknown origin) assessed as inhibition constant in presence of ATPMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity to EGFR-D770-N771insNPG mutant (unknown origin) assessed as inhibition constant in presence of ATPMore data for this Ligand-Target Pair
