Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50020448
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629961(CHEMBL5406585)
Affinity DataIC50: 4.20nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629968(CHEMBL5404986)
Affinity DataIC50: 4.80nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629963(CHEMBL5416229)
Affinity DataIC50: 12nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629970(CHEMBL5395771)
Affinity DataIC50: 15nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629953(CHEMBL5438588)
Affinity DataIC50: 16nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629970(CHEMBL5395771)
Affinity DataIC50: 19nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD2-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629962(CHEMBL5430730)
Affinity DataIC50: 19nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50380682(CHEMBL2017291 | I-BET151 (16))
Affinity DataIC50: 25nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629965(CHEMBL5405536)
Affinity DataIC50: 25nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629970(CHEMBL5395771)
Affinity DataIC50: 25nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD3-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629957(CHEMBL5400407)
Affinity DataIC50: 32nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629956(CHEMBL5422966)
Affinity DataIC50: 38nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629969(CHEMBL5427136)
Affinity DataIC50: 39nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629966(CHEMBL5411662)
Affinity DataIC50: 42nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629967(CHEMBL5432892)
Affinity DataIC50: 45nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629964(CHEMBL5432627)
Affinity DataIC50: 50nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629970(CHEMBL5395771)
Affinity DataIC50: 55nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from BRD4-BD2 (unknown origin) incubated for 3 hrs by HTRF based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629954(CHEMBL5399062)
Affinity DataIC50: 61nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629970(CHEMBL5395771)
Affinity DataIC50: 68nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRDT-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629970(CHEMBL5395771)
Affinity DataIC50: 81nMAssay Description:Inhibition of NanoLuc-tagged full length BRD4 (unknown origin) transfected in HEK293 cells coexpressing histone H4-halo-tagged fusion vector preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629955(CHEMBL5413739)
Affinity DataIC50: 94nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629960(CHEMBL5403013)
Affinity DataIC50: 112nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629958(CHEMBL5414236)
Affinity DataIC50: 122nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Maruho Co.

Curated by ChEMBL
LigandPNGBDBM50629959(CHEMBL5421597)
Affinity DataIC50: 157nMAssay Description:Displacement of Biotin-tagged [Lys(5,8,12,16)Ac]H4(1 to 21) peptide from GST-tagged BRD4-BD1 (unknown origin) incubated for 3 hrs by HTRF based TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed