Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50020269
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM349662(2-{[4-(6-{[(4-cyano-2-fluorophenyl)(methyl-d2)]oxy...)
Affinity DataEC50:  13nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628333(CHEMBL5414345)
Affinity DataEC50:  35nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628334(CHEMBL5419346)
Affinity DataEC50:  32nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628335(CHEMBL5434776)
Affinity DataEC50:  19nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628336(CHEMBL5396298)
Affinity DataEC50:  15nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628337(CHEMBL5399359)
Affinity DataEC50:  15nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628338(CHEMBL5429544)
Affinity DataEC50:  14nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628339(CHEMBL5440900)
Affinity DataEC50:  5.80nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50628340(CHEMBL5418836)
Affinity DataEC50:  4.10nMAssay Description:Displacement of [125I]-GLP1 from GLP-1 receptor (unknown origin) expressed in CHO cells membrane pre-incubated for 10 mins followed by [125I]-GLP1 ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed