Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50020238
TargetBromodomain-containing protein 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50628038(CHEMBL5428113)
Affinity DataKi:  680nMAssay Description:Binding affinity to human recombinant BRD4BD1 (44 to 168 residues) expressed in Escherichia coli BL23 (DE3) by fluorescence polarization analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50628037(CHEMBL5416132)
Affinity DataKi:  760nMAssay Description:Binding affinity to human recombinant BRD4BD1 (44 to 168 residues) expressed in Escherichia coli BL23 (DE3) by fluorescence polarization analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50628036(CHEMBL5431735)
Affinity DataKi:  910nMAssay Description:Binding affinity to human recombinant BRD4BD1 (44 to 168 residues) expressed in Escherichia coli BL23 (DE3) by fluorescence polarization analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50628036(CHEMBL5431735)
Affinity DataKi:  1.44E+3nMAssay Description:Binding affinity to human recombinant BRD4BD2 (333 to 460 residues) expressed in Escherichia coli BL23 (DE3) by fluorescence polarization analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50628037(CHEMBL5416132)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human recombinant BRD4BD2 (333 to 460 residues) expressed in Escherichia coli BL23 (DE3) by fluorescence polarization analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50628038(CHEMBL5428113)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity to human recombinant BRD4BD2 (333 to 460 residues) expressed in Escherichia coli BL23 (DE3) by fluorescence polarization analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed