Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50020009
TargetAngiopoietin-1 receptor(Human)
University of South China

Curated by ChEMBL
LigandPNGBDBM50625562(CHEMBL5401507)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
University of South China

Curated by ChEMBL
LigandPNGBDBM21079(1-[4-(3-azanyl-1H-indazol-4-yl)phenyl]-3-(2-fluora...)
Affinity DataIC50: 8nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of South China

Curated by ChEMBL
LigandPNGBDBM21079(1-[4-(3-azanyl-1H-indazol-4-yl)phenyl]-3-(2-fluora...)
Affinity DataIC50: 28nMAssay Description:Inhibition of KDR (unknown origin) using biotin as substrate preincubated for 1 hr in presence of ATP and measured after 1 hr by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of South China

Curated by ChEMBL
LigandPNGBDBM50625562(CHEMBL5401507)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human VEGFRMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
University of South China

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of VEGFR2 in HUVEC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
University of South China

Curated by ChEMBL
LigandPNGBDBM50625561(CHEMBL5422319)
Affinity DataIC50: 7.32E+4nMAssay Description:Inhibition of VEGFR2 in HUVEC cellsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed