Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50019896
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624358(CHEMBL5403275)
Affinity DataEC50:  920nMAssay Description:Inhibition of interaction of PD-1 (unknown origin) expressed in Jurkat T cells carrying luciferase reporter under the control of NFAT promoter/PD-L1 ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Human)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624358(CHEMBL5403275)
Affinity DataKd:  44nMAssay Description:Binding affinity to human PD-L1 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624358(CHEMBL5403275)
Affinity DataKd:  218nMAssay Description:Binding affinity to mouse PD-L1 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProgrammed cell death 1 ligand 1(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624358(CHEMBL5403275)
Affinity DataKd:  438nMAssay Description:Binding affinity to mouse PD-L1 assessed as dissociation constant by MST analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624364(CHEMBL4802680)
Affinity DataEC50:  4.65E+3nMAssay Description:Inhibition of interaction of PD-1 (unknown origin) expressed in Jurkat T cells carrying luciferase reporter under the control of NFAT promoter/PD-L1 ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM575481(US11459339, Example 1 | N,N′-(2,2′-dim...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50239948(US9850225, Example 1166 | CHEMBL4071326)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624358(CHEMBL5403275)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of GST-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) interaction by HTRF binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50580548(CHEMBL5081629)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624359(CHEMBL5435574)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of GST-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) interaction by HTRF binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50581932(CHEMBL5093206)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624360(CHEMBL5432440)
Affinity DataIC50: 4nMAssay Description:Inhibition of GST-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) interaction by HTRF binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624363(CHEMBL5397551)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of GST-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) interaction by HTRF binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50578293(CHEMBL4873960)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624365(CHEMBL5423998)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624362(CHEMBL5402633)
Affinity DataIC50: 11nMAssay Description:Inhibition of GST-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) interaction by HTRF binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50624361(CHEMBL5420228)
Affinity DataIC50: 12nMAssay Description:Inhibition of GST-tagged PD-1 (unknown origin)/His-tagged PD-L1 (unknown origin) interaction by HTRF binding assay relative to controlMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50239947(US9872852, Example 202 | CHEMBL4089730 | US2023030...)
Affinity DataIC50: 18nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Zunyi Medical University

Curated by ChEMBL
LigandPNGBDBM50550710(CHEMBL4749782)
Affinity DataIC50: 133nMAssay Description:Inhibition of PD-1 (unknown origin)/PD-L1 (unknown origin) interaction by HTRF binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed