Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50019570
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542856(CHEMBL4639709)
Affinity DataEC50:  170nMAssay Description:Agonist potency at human Y4 receptor expressed in HEK293T-NlucN-mGSi/Y4R-NlucC cells by miniGsi protein recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578268(CHEMBL4856311)
Affinity DataEC50:  1nMAssay Description:Agonist potency at human Y4 receptor expressed in HEK293T-NlucN-mGSi/Y4R-NlucC cells by miniGsi protein recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578262(CHEMBL4873376)
Affinity DataEC50:  1.70nMAssay Description:Agonist potency at human Y4 receptor expressed in HEK293T-NlucN-mGSi/Y4R-NlucC cells by miniGsi protein recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620622(CHEMBL5418083)
Affinity DataEC50:  610nMAssay Description:Agonist potency at human Y4 receptor expressed in HEK293T-NlucN-mGSi/Y4R-NlucC cells by miniGsi protein recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620621(CHEMBL5426658)
Affinity DataEC50:  20nMAssay Description:Agonist potency at human Y4 receptor expressed in HEK293T-NlucN-mGSi/Y4R-NlucC cells by miniGsi protein recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542834(CHEMBL4633593)
Affinity DataEC50:  110nMAssay Description:Agonist potency at human Y4 receptor expressed in HEK293T-NlucN-mGSi/Y4R-NlucC cells by miniGsi protein recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578268(CHEMBL4856311)
Affinity DataKi:  0.0330nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50578262(CHEMBL4873376)
Affinity DataKi:  0.0480nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620621(CHEMBL5426658)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542856(CHEMBL4639709)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542834(CHEMBL4633593)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620622(CHEMBL5418083)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620621(CHEMBL5426658)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]UR-MK299 from human Y1 receptor expressed in human SK-N-MC cells measured after 90 mins by MicroBeta plate counter based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620623(CHEMBL5431678)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620624(CHEMBL5434829)
Affinity DataKi:  910nMAssay Description:Displacement of [3H]UR-KK200 from human Y4 receptor expressed in CHO-Gqi5-mtAQE cells measured after 90 mins by MicroBeta plate counter based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620621(CHEMBL5426658)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y2 receptor expressed in CHO cells measured after 90 mins by MicroBeta plate counter based competition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620623(CHEMBL5431678)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]UR-MK299 from human Y1 receptor expressed in human SK-N-MC cells measured after 90 mins by MicroBeta plate counter based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620623(CHEMBL5431678)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y5 receptor expressed in HEC-1B cells measured after 90 mins by MicroBeta plate counter based competiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620624(CHEMBL5434829)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y5 receptor expressed in HEC-1B cells measured after 90 mins by MicroBeta plate counter based competiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620624(CHEMBL5434829)
Affinity DataKi: >1.05E+3nMAssay Description:Displacement of [3H]UR-MK299 from human Y1 receptor expressed in human SK-N-MC cells measured after 90 mins by MicroBeta plate counter based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542834(CHEMBL4633593)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]UR-MK299 from human Y1 receptor expressed in human SK-N-MC cells measured after 90 mins by MicroBeta plate counter based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620624(CHEMBL5434829)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y2 receptor expressed in CHO cells measured after 90 mins by MicroBeta plate counter based competition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620623(CHEMBL5431678)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y2 receptor expressed in CHO cells measured after 90 mins by MicroBeta plate counter based competition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620622(CHEMBL5418083)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y2 receptor expressed in CHO cells measured after 90 mins by MicroBeta plate counter based competition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetP2Y purinoceptor 1(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620622(CHEMBL5418083)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]UR-MK299 from human Y1 receptor expressed in human SK-N-MC cells measured after 90 mins by MicroBeta plate counter based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620621(CHEMBL5426658)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y5 receptor expressed in HEC-1B cells measured after 90 mins by MicroBeta plate counter based competiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50620622(CHEMBL5418083)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y5 receptor expressed in HEC-1B cells measured after 90 mins by MicroBeta plate counter based competiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542834(CHEMBL4633593)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y2 receptor expressed in CHO cells measured after 90 mins by MicroBeta plate counter based competition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetNeuropeptide Y receptor type 5(Human)
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50542834(CHEMBL4633593)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]propionyl-pNPY from human Y5 receptor expressed in HEC-1B cells measured after 90 mins by MicroBeta plate counter based competiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed