Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50020257
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50104413(Glutamyl-gamma-boronate analogue | CHEMBL87796)
Affinity DataKi:  5nMAssay Description:Inhibition of GGT1 (unknown origin) transpeptidation assessed as inhibition constant using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50104413(Glutamyl-gamma-boronate analogue | CHEMBL87796)
Affinity DataKi:  25nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628182(CHEMBL5400857)
Affinity DataKi:  920nMAssay Description:Inhibition of GGT1 (unknown origin) transpeptidation assessed as inhibition constant using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628182(CHEMBL5400857)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628187(CHEMBL1492424)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of GGT1 (unknown origin) transpeptidation assessed as inhibition constant using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628184(CHEMBL5405005)
Affinity DataKi:  1.98E+5nMAssay Description:Inhibition of GGT1 (unknown origin) transpeptidation assessed as inhibition constant using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628187(CHEMBL1492424)
Affinity DataKi:  3.76E+5nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628183(CHEMBL5397333)
Affinity DataKi:  4.44E+5nMAssay Description:Inhibition of GGT1 (unknown origin) transpeptidation assessed as inhibition constant using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628184(CHEMBL5405005)
Affinity DataKi:  7.03E+5nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628183(CHEMBL5397333)
Affinity DataKi:  8.74E+5nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628185(CHEMBL5406958)
Affinity DataKi: >4.00E+6nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628186(CHEMBL5404531)
Affinity DataKi: >5.00E+6nMAssay Description:Inhibition of GGT1 (unknown origin) assessed as GSH hydrolysis by measuring inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50628185(CHEMBL5406958)
Affinity DataKi:  3.82E+6nMAssay Description:Inhibition of GGT1 (unknown origin) transpeptidation assessed as inhibition constant using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed