Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50020252
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM81395(APO-866 | US20240327418, Example FK866 | US2024030...)
Affinity DataIC50: 0.560nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628141(CHEMBL5408614)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628148(CHEMBL5401142)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628144(CHEMBL5398077)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628145(CHEMBL5432491)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628142(CHEMBL5404254)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628146(CHEMBL5428751)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628143(CHEMBL5394343)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Changzhou University

Curated by ChEMBL
LigandPNGBDBM50628147(CHEMBL5408297)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed