Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019545
TargetSuccinate receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620363(CHEMBL5439297)
Affinity DataKd:  1.58E+3nMAssay Description:Binding affinity to N-terminal Nluc-tagged human succinate receptor 1 expressed in human Flp-In-T-REx-293 cells using assessed as dissociation consta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620364(CHEMBL5438140)
Affinity DataKd:  990nMAssay Description:Binding affinity to N-terminal Nluc-tagged human succinate receptor 1 expressed in human Flp-In-T-REx-293 cells using assessed as dissociation consta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Mus musculus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620363(CHEMBL5439297)
Affinity DataKd:  1.16E+3nMAssay Description:Binding affinity to N-terminal Nluc-tagged mouse succinate receptor 1 expressed in human Flp-In-T-REx-293 cells using assessed as dissociation consta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Mus musculus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620364(CHEMBL5438140)
Affinity DataKd:  1.17E+3nMAssay Description:Binding affinity to N-terminal Nluc-tagged mouse succinate receptor 1 expressed in human Flp-In-T-REx-293 cells using assessed as dissociation consta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620365(CHEMBL5399663)
Affinity DataKd:  310nMAssay Description:Binding affinity to N-terminal Nluc-tagged human succinate receptor 1 expressed in Flp-In-T-REx-293 cells assessed as dissociation constant incubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620364(CHEMBL5438140)
Affinity DataKd:  620nMAssay Description:Binding affinity to N-terminal Nluc-tagged human succinate receptor 1 expressed in human Flp-In-T-REx-293 cells assessed as dissociation constant inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620365(CHEMBL5399663)
Affinity DataKd:  560nMAssay Description:Binding affinity to N-terminal Nluc-tagged human succinate receptor 1 expressed in human Flp-In-T-REx-293 cells assessed as dissociation constant inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetSuccinate receptor 1(Mus musculus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50620364(CHEMBL5438140)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to N-terminal Nluc-tagged mouse succinate receptor 1 expressed in human Flp-In-T-REx-293 cells assessed as dissociation constant inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed