Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50019256
TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50617206(CHEMBL5439289)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM552651(WO2022101377, Example 50)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM552674(WO2022101377, Example 73)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50617208(CHEMBL5411707)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50617205(CHEMBL5413888)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50617207(CHEMBL5400532)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed