Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50018859
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM45440(4-[5-(4-carbamimidoylphenoxy)pentoxy]benzenecarbox...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TMPRSS2 (247 to 492 residues) (unknown origin) peptidase domain expressed in Escherichia coli BL21 (DE3) incubated for 30 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613302(CHEMBL5285196)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613298(CHEMBL5270157)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613303(CHEMBL5266850)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50368092(GNF-PF-3839 | PROPAMIDINE CHLORIDE)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of TMPRSS2 (247 to 492 residues) (unknown origin) peptidase domain expressed in Escherichia coli BL21 (DE3) incubated for 30 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613299(CHEMBL5271456)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613305(CHEMBL5287275)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613300(CHEMBL5275059)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613301(CHEMBL5270536)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613304(CHEMBL5275526)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50122613(3,4-dihydroisoquinoline-2(1H)-carboximidamide | De...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of TMPRSS2 (106 to 492 residues) (unknown origin) using Boc-QAR-AMC as substrate measured for 20 mins by spectrophotometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetTransmembrane protease serine 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50122613(3,4-dihydroisoquinoline-2(1H)-carboximidamide | De...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of TMPRSS2 (247 to 492 residues) (unknown origin) peptidase domain expressed in Escherichia coli BL21 (DE3) incubated for 30 mins followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed