Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50020424
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629819(CHEMBL5406096)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629817(CHEMBL5402946)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 40...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629820(CHEMBL5401982)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629814(CHEMBL5395799)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629811(CHEMBL5434226)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629815(CHEMBL5413257)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629821(CHEMBL5428297)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 40...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629812(CHEMBL5406836)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 60...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 60...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629822(CHEMBL5424305)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 40...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629813(CHEMBL5418350)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 8.10nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 60...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 40...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50469180(CHEMBL4292755)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629810(CHEMBL5420802)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50277584(N-(5-methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629818(CHEMBL5410160)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using STK-substrate 2-biotin as substrate incubated for 60...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629823(CHEMBL5435989)
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetAurora kinase A(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50629816(CHEMBL5398559)
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human Aurora A (1 to 403 residues) expressed in Escherichia coli using FAM-labeled peptide as substrate preincubated for 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed