Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 50019688
Affinity DataEC50: 158nMAssay Description:Agonist activity at human CB2 receptor stably expressed in CHO-K1 cells co-expressing Galphaq16 by Fluo-4AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 244nMAssay Description:Agonist activity at human CB2 receptor stably expressed in CHO-K1 cells co-expressing Galphaq16 by Fluo-4AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 7.71E+3nMAssay Description:Agonist activity at human CB2 receptor stably expressed in CHO-K1 cells co-expressing Galphaq16 by Fluo-4AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 1.30E+3nMAssay Description:Agonist activity at human CB2 receptor stably expressed in CHO-K1 cells co-expressing Galphaq16 by Fluo-4AM dye based calcium mobilization assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 0.630nMAssay Description:Agonist activity at human CB2 receptor stably expressed in HEK293 cells assessed as induction of beta-arrestin 2 recruitment incubated for 2 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at human CB2 receptor stably expressed in HEK293 cells assessed as induction of beta-arrestin 2 recruitment incubated for 2 hrs by l...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 82nMAssay Description:Agonist activity at human CB2 receptor stably expressed in HEK293 cells assessed as induction of beta-arrestin 2 recruitment incubated for 2 hrs by l...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]CP55940 from rat brain membrane CB1 receptor incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 150nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 152nMAssay Description:Pseudo-irreversible inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellm...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 304nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 390nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 580nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 620nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 711nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 780nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 810nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.01E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.02E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.06E+3nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.19E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.35E+3nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.78E+3nMAssay Description:Inhibition of human BChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.21E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.90E+3nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 3.46E+3nMAssay Description:Pseudo-irreversible inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellm...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 3.58E+3nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 to 60 mins followed by substrate addition by spectrophotometric...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 3.85E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 4.02E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 4.22E+3nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 4.50E+3nMAssay Description:Pseudo-irreversible inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellm...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 5.53E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membrane incubated for 3 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 8.66E+3nMAssay Description:Pseudo-irreversible inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellm...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 9.01E+3nMAssay Description:Pseudo-irreversible inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellm...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.00E+4nMAssay Description:Pseudo-irreversible inhibition of human BChE using butyrylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ell...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Pseudo-irreversible inhibition of human AChE using acetylthiocholine iodide as substrate incubated for 20 mins followed by substrate addition by Ellm...More data for this Ligand-Target Pair








3D Structure (crystal)















