Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50018957
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614167(CHEMBL5288335)
Affinity DataIC50: 6nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165363(US9062043, Table 20b, Compound 21 | US9062043, Tab...)
Affinity DataIC50: 17nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614175(CHEMBL5283179)
Affinity DataIC50: 19nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165347(US9062043, Table 20b, Compound 9 | US9062043, Tabl...)
Affinity DataIC50: 19nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614173(CHEMBL5289971)
Affinity DataIC50: 19nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614167(CHEMBL5288335)
Affinity DataIC50: 21nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614172(CHEMBL5287614)
Affinity DataIC50: 22nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614168(CHEMBL5277426)
Affinity DataIC50: 25nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165350(US9062043, Table 20b, Compound 11 | US9062043, Tab...)
Affinity DataIC50: 34nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614175(CHEMBL5283179)
Affinity DataIC50: 36nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614169(CHEMBL5288569)
Affinity DataIC50: 42nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165341(US9062043, Table 20b, Compound 5 | US9062043, Tabl...)
Affinity DataIC50: 43nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165353(US9062043, Table 20b, Compound 14 | US9062043, Tab...)
Affinity DataIC50: 51nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165364(US9062043, Table 20b, Compound 22 | US9062043, Tab...)
Affinity DataIC50: 62nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614170(CHEMBL5273686)
Affinity DataIC50: 63nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50566496(CHEMBL4846181)
Affinity DataIC50: 66nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614164(CHEMBL5273101)
Affinity DataIC50: 93nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614172(CHEMBL5287614)
Affinity DataIC50: 100nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165347(US9062043, Table 20b, Compound 9 | US9062043, Tabl...)
Affinity DataIC50: 110nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614171(CHEMBL5279015)
Affinity DataIC50: 110nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165359(US9062043, Table 20b, Compound 18 | US9062043, Tab...)
Affinity DataIC50: 130nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614165(CHEMBL5272174)
Affinity DataIC50: 140nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614173(CHEMBL5289971)
Affinity DataIC50: 150nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165349(US9062043, Table 20b, Compound 10 | US9062043, Tab...)
Affinity DataIC50: 180nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50: 180nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 200nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165341(US9062043, Table 20b, Compound 5 | US9062043, Tabl...)
Affinity DataIC50: 220nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165363(US9062043, Table 20b, Compound 21 | US9062043, Tab...)
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50: 240nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614168(CHEMBL5277426)
Affinity DataIC50: 240nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165350(US9062043, Table 20b, Compound 11 | US9062043, Tab...)
Affinity DataIC50: 260nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614166(CHEMBL5284276)
Affinity DataIC50: 270nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614169(CHEMBL5288569)
Affinity DataIC50: 300nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165364(US9062043, Table 20b, Compound 22 | US9062043, Tab...)
Affinity DataIC50: 300nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165340(US9062043, Table 20b, Compound 4 | US9062043, Tabl...)
Affinity DataIC50: 340nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165353(US9062043, Table 20b, Compound 14 | US9062043, Tab...)
Affinity DataIC50: 350nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50566496(CHEMBL4846181)
Affinity DataIC50: 350nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165207(US9062043, Table 13, Compound 1 | US9062043, Table...)
Affinity DataIC50: 420nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165359(US9062043, Table 20b, Compound 18 | US9062043, Tab...)
Affinity DataIC50: 430nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165362(US9062043, Table 13, Compound 29 | US8168651, Comp...)
Affinity DataIC50: 450nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614171(CHEMBL5279015)
Affinity DataIC50: 550nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614164(CHEMBL5273101)
Affinity DataIC50: 570nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165349(US9062043, Table 20b, Compound 10 | US9062043, Tab...)
Affinity DataIC50: 680nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614170(CHEMBL5273686)
Affinity DataIC50: 740nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614165(CHEMBL5272174)
Affinity DataIC50: 830nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 920nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614166(CHEMBL5284276)
Affinity DataIC50: 930nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50614163(CHEMBL5288779)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of wild type human CK2alpha' in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165362(US9062043, Table 13, Compound 29 | US8168651, Comp...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM165340(US9062043, Table 20b, Compound 4 | US9062043, Tabl...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
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