Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50018956
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614160(CHEMBL5271690)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant human furin using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614159(CHEMBL5275267)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant human furin using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614158(CHEMBL5276332)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant human furin using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614161(CHEMBL5285236)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human furin using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614160(CHEMBL5271690)
Affinity DataKi:  0.210nMAssay Description:Inhibition of recombinant human furin assessed as inhibition constant using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614159(CHEMBL5275267)
Affinity DataKi:  0.25nMAssay Description:Inhibition of recombinant human furin assessed as inhibition constant using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614158(CHEMBL5276332)
Affinity DataKi:  0.270nMAssay Description:Inhibition of recombinant human furin assessed as inhibition constant using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614161(CHEMBL5285236)
Affinity DataKi:  0.380nMAssay Description:Inhibition of recombinant human furin assessed as inhibition constant using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFurin(Human)
University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50614162(CHEMBL5277422)
Affinity DataKi:  0.490nMAssay Description:Inhibition of recombinant human furin assessed as inhibition constant using Pyr-Arg-Thr-Lys-Arg-AMC as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed