Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50020164
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50029464(LY-292728 | 5-(2-Carboxy-ethyl)-6-[3-(5-ethyl-4'-f...)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity against LTB4 receptor in human Neutrophil incubated for 10 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627055(CHEMBL5431150)
Affinity DataIC50: 12nMAssay Description:Antagonist activity against LTB4 receptor in human Neutrophil incubated for 10 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627050(CHEMBL5425581)
Affinity DataIC50: 288nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50001610(CHEMBL14823 | CGS 24115 | 7-[3-(4-Acetyl-3-methoxy...)
Affinity DataIC50: 300nMAssay Description:Antagonist activity against LTB4 receptor in human Neutrophil incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627051(CHEMBL5425438)
Affinity DataIC50: 439nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627052(CHEMBL5404528)
Affinity DataIC50: 477nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627054(CHEMBL5408842)
Affinity DataIC50: 710nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627049(CHEMBL5440367)
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627053(CHEMBL5411386)
Affinity DataIC50: 5.61E+3nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627048(CHEMBL5424341)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against LTB4 receptor in human U-937 cells incubated for 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50627056(CHEMBL5428366)
Affinity DataKi:  1nMAssay Description:Antagonist activity against LTB4 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50037390(3-{(S)-2-(2-Carboxy-ethyl)-7-[3-(2-cyclopropylmeth...)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity against LTB4 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50001609(CHEMBL328712 | 8-Benzyloxy-4-[(methyl-phenethyl-ca...)
Affinity DataKi:  2nMAssay Description:Antagonist activity against LTB4 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Sultan Moulay Slimane University

Curated by ChEMBL
LigandPNGBDBM50037382(ONO 4057 | 5-{2-(2-Carboxy-ethyl)-3-[6-(4-methoxy-...)
Affinity DataKi:  4nMAssay Description:Antagonist activity against LTB4 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed