Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50020156
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetHistamine H1 receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50079527(CHEMBL101740 | cis-doxepin | DOXEPIN | (3E)-3-dibe...)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]-Pyrilamine from human histamine H1 expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50581210(Ipratropium | Ipratropium cation | Ipratropium ion...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-Pirenzepine from human muscarinic M1 expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C expressed in HeLa cells membrane incubated for 1 hr by microbeta liquid scintillation counting ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626918(CHEMBL5404031)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626907(CHEMBL5415412)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626919(CHEMBL5412886)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626915(CHEMBL5424052)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626907(CHEMBL5415412)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626918(CHEMBL5404031)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626919(CHEMBL5412886)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626917(CHEMBL5422196)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626916(CHEMBL5435580)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626908(CHEMBL5409227)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626917(CHEMBL5422196)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626912(CHEMBL5429491)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626912(CHEMBL5429491)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626909(CHEMBL5395668)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626920(CHEMBL5432478)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626914(CHEMBL5431642)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626914(CHEMBL5431642)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626906(CHEMBL5398291)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626913(CHEMBL5411002)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetHistamine H1 receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626908(CHEMBL5409227)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-Pyrilamine from human histamine H1 expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626908(CHEMBL5409227)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626916(CHEMBL5435580)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626908(CHEMBL5409227)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C expressed in HeLa cells membrane incubated for 1 hr by microbeta liquid scintillation counting ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626915(CHEMBL5424052)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626920(CHEMBL5432478)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626908(CHEMBL5409227)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626906(CHEMBL5398291)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626911(CHEMBL5439203)
Affinity DataKi:  139nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626917(CHEMBL5422196)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626920(CHEMBL5432478)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626916(CHEMBL5435580)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626918(CHEMBL5404031)
Affinity DataKi:  179nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626912(CHEMBL5429491)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626906(CHEMBL5398291)
Affinity DataKi:  216nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626909(CHEMBL5395668)
Affinity DataKi:  239nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626913(CHEMBL5411002)
Affinity DataKi:  243nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626911(CHEMBL5439203)
Affinity DataKi:  264nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626913(CHEMBL5411002)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626919(CHEMBL5412886)
Affinity DataKi:  318nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626907(CHEMBL5415412)
Affinity DataKi:  321nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626909(CHEMBL5395668)
Affinity DataKi:  401nMAssay Description:Displacement of [3H]-ketanserin from human 5-HT2A receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626910(CHEMBL5420627)
Affinity DataKi:  405nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A receptor expressed in HEK293 cells membrane incubated for 1 hr by microbeta liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626914(CHEMBL5431642)
Affinity DataKi:  552nMAssay Description:Displacement of [3H]-Mesulergine from human 5-HT2C expressed in HeLa cells membrane incubated for 1 hr by microbeta liquid scintillation counting ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetD(2) dopamine receptor(Human)
Medical University of Lublin

Curated by ChEMBL
LigandPNGBDBM50626910(CHEMBL5420627)
Affinity DataKi:  557nMAssay Description:Displacement of [3H]-spiperone from human D2s receptor expressed in CHO-K1 cells membrane incubated for 1 hr by microbeta liquid scintillation counti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
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