Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50020685
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632703(CHEMBL5424187)
Affinity DataIC50: 1nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632695(CHEMBL5404620)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632707(CHEMBL5397693)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632709(CHEMBL5412884)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632708(CHEMBL5411391)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50203882(2-methyl-N-{4-[1-(4-methyl-piperazine-1-carbonyl)-...)
Affinity DataIC50: 4nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632700(CHEMBL5399936)
Affinity DataIC50: 4nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632699(CHEMBL5404280)
Affinity DataIC50: 6nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632701(CHEMBL5412094)
Affinity DataIC50: 6nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632696(CHEMBL5400674)
Affinity DataIC50: 13nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632694(CHEMBL5400852)
Affinity DataIC50: 14nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632674(CHEMBL5407071)
Affinity DataIC50: 24nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632713(CHEMBL5434812)
Affinity DataIC50: 26nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632698(CHEMBL5400080)
Affinity DataIC50: 27nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632711(CHEMBL5412408)
Affinity DataIC50: 28nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632690(CHEMBL5399315)
Affinity DataIC50: 29nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632712(CHEMBL5410064)
Affinity DataIC50: 33nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632697(CHEMBL5437244)
Affinity DataIC50: 33nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632674(CHEMBL5407071)
Affinity DataIC50: 34nMAssay Description:Inhibition of CCR8-mediated cell migration in CCL1-induced human PBMC preincubated for 1 hr followed by CCL1 addition measured after 4 hrs by cell co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632710(CHEMBL5402712)
Affinity DataIC50: 37nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632705(CHEMBL5397155)
Affinity DataIC50: 46nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632715(CHEMBL5434069)
Affinity DataIC50: 79nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632692(CHEMBL5395905)
Affinity DataIC50: 85nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632720(CHEMBL5432261)
Affinity DataIC50: 85nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632714(CHEMBL5438933)
Affinity DataIC50: 90nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632688(CHEMBL5432566)
Affinity DataIC50: 112nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632717(CHEMBL5437230)
Affinity DataIC50: 129nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632702(CHEMBL5435573)
Affinity DataIC50: 158nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632716(CHEMBL5394357)
Affinity DataIC50: 200nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632721(CHEMBL5432453)
Affinity DataIC50: 251nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632691(CHEMBL5424675)
Affinity DataIC50: 303nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632687(CHEMBL5415778)
Affinity DataIC50: 500nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632706(CHEMBL5415309)
Affinity DataIC50: 735nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632676(CHEMBL5420573)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632722(CHEMBL5422825)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632719(CHEMBL5398519)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632693(CHEMBL5418685)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632718(CHEMBL5437085)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632675(CHEMBL5405169)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632677(CHEMBL5422913)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632678(CHEMBL5434367)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632679(CHEMBL5420476)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632680(CHEMBL5399791)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632681(CHEMBL5417132)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632682(CHEMBL5406553)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632704(CHEMBL5428200)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632683(CHEMBL5423271)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632684(CHEMBL5425376)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632685(CHEMBL5418858)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632686(CHEMBL5437965)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
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