Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50020658
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50632389(CHEMBL5414494)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to wild type SARS-COV2 main protease expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by small angle X-ray...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50632389(CHEMBL5414494)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to SARS-COV2 main protease assessed as dissociation constant by analytical ultracentrifugation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetReplicase polyprotein 1ab(2019-nCoV)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50632389(CHEMBL5414494)
Affinity DataKd:  140nMAssay Description:Binding affinity to SARS-COV2 main protease assessed as dissociation constant by mass spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed