Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50020137
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM168025(US9073926, 59)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of RSK2 (unknown origin) preincubated for 1 hr followed by substrate addition and measured after 1 hr by luciferase analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360301(CHEMBL1933288 | US9150577, 93)
Affinity DataIC50: 1nMAssay Description:Inhibition of human RSK2 in MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360291(CHEMBL1933278 | US9150577, 114)
Affinity DataIC50: 2nMAssay Description:Inhibition of human RSK2 in MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360296(CHEMBL1933283 | US9150577, 96)
Affinity DataIC50: 12nMAssay Description:Inhibition of human RSK2 in MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50248765(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)
Affinity DataIC50: 15nMAssay Description:Inhibition of wild type RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50248767(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)
Affinity DataIC50: 15nMAssay Description:Inhibition of wild type RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360299(CHEMBL1933286 | US9150577, 54)
Affinity DataIC50: 20nMAssay Description:Inhibition of human RSK2 in MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50426389(CHEMBL2321925)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant His-tagged RSK2 (unknown origin) expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50360298(CHEMBL1933285 | US9150577, 53)
Affinity DataIC50: 20nMAssay Description:Inhibition of human RSK2 in MCF7 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50241294(kaempferol-3-O-(3,4-di-O-acetyl-alpha-L-rhamnopyra...)
Affinity DataIC50: 89nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM8296(CHEMBL102714 | cid_176158 | 3-(2,4-dichlorophenyl)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50166289(CHEBI:43645 | CHEMBL216543)
Affinity DataIC50: 100nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM3175(Bisindolylmaleimide 11b | Ro 31-8220 | CHEMBL6291 ...)
Affinity DataIC50: 200nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626653(CHEMBL5419696)
Affinity DataIC50: 440nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM2683(2-[1-(3-dimethylaminopropyl)-indol-3-yl]-3-(indol-...)
Affinity DataIC50: 610nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626654(CHEMBL5401630)
Affinity DataIC50: 870nMAssay Description:Inhibition of recombinant His-tagged RSK2 (unknown origin) expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626655(CHEMBL5439691)
Affinity DataIC50: 870nMAssay Description:Inhibition of recombinant His-tagged RSK2 (unknown origin) expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM7457(2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-chromen-4-on...)
Affinity DataIC50: 891nMAssay Description:Inhibition of RSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626652(CHEMBL4303592)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of RSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626652(CHEMBL4303592)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50241294(kaempferol-3-O-(3,4-di-O-acetyl-alpha-L-rhamnopyra...)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM7462(cid_5280863 | CHEMBL150 | 3,5,7-trihydroxy-2-(4-hy...)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of RSK2 expressed in human MCF7 cells incubated for 1 hrs byMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50343656(5-(2-(4-hydroxyphenyl)hydrazono)pyrimidine-2,4,6(1...)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50384788(LAPACHOL)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM241958(5-(2-(4-Hydroxyphenyl)hydrazono)-dihydro-2-thioxop...)
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of human RSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626652(CHEMBL4303592)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM7457(2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-chromen-4-on...)
Affinity DataIC50: 2.78E+3nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM7457(2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-chromen-4-on...)
Affinity DataIC50: 3.79E+3nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 4.42E+3nMAssay Description:Inhibition of RSK2 expressed in human MCF7 cells incubated for 1 hrs byMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50325671(CHEMBL8996 | eriodicryol | (S)-2-(3,4-dihydroxyphe...)
Affinity DataIC50: 4.77E+3nMAssay Description:Inhibition of RSK2 expressed in human MCF7 cells incubated for 1 hrs byMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-6(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50626656(CHEMBL5418355)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50504654(CHEBI:76004 | AZL 0 211089 | AZL O 211089 | AZL-02...)
Affinity DataIC50: 2.25E+5nMAssay Description:Inhibition of human recombinant RSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed