Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50020757
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633339(CHEMBL5404184)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633344(CHEMBL5418688)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633356(CHEMBL5410721)
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633342(CHEMBL5410158)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633338(CHEMBL5436718)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633349(CHEMBL5426884)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633353(CHEMBL5437483)
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633336(CHEMBL5421814)
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633343(CHEMBL5421760)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633340(CHEMBL5436602)
Affinity DataIC50: 5.38E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633346(CHEMBL5407982)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633352(CHEMBL5407966)
Affinity DataIC50: 5.55E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633345(CHEMBL5412577)
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633347(CHEMBL5420345)
Affinity DataIC50: 5.75E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633355(CHEMBL5416119)
Affinity DataIC50: 5.76E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633341(CHEMBL5426350)
Affinity DataIC50: 6.23E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633351(CHEMBL5407902)
Affinity DataIC50: 6.29E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633357(CHEMBL5424970)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633350(CHEMBL5433909)
Affinity DataIC50: 6.45E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633358(CHEMBL2043176)
Affinity DataIC50: 6.98E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633348(CHEMBL5426575)
Affinity DataIC50: 8.09E+3nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633354(CHEMBL5438109)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHypoxia-inducible factor 1-alpha inhibitor(Human)
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633337(CHEMBL5414621)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of HIF-1 alpha transcriptional activity in human U-251 cells incubated for 24 hrs under hypoxia condition by luciferse reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed