Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50019238
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617034(CHEMBL5419363)
Affinity DataIC50: 1nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617027(CHEMBL5436066)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617014(CHEMBL5434556)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617015(CHEMBL5434041)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617016(CHEMBL5432825)
Affinity DataIC50: 3nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617017(CHEMBL5431304)
Affinity DataIC50: 5nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617021(CHEMBL5408520)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617013(CHEMBL5427802)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617030(CHEMBL5393990)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617024(CHEMBL5404212)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617022(CHEMBL5426154)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617020(CHEMBL5395872)
Affinity DataIC50: 12nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617028(CHEMBL5417707)
Affinity DataIC50: 12nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617023(CHEMBL5436593)
Affinity DataIC50: 16nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 23nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 26nMAssay Description:Inhibition of BRD2-BD1/2 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617014(CHEMBL5434556)
Affinity DataIC50: 31nMAssay Description:Inhibition of BRD2-BD1/2 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617014(CHEMBL5434556)
Affinity DataIC50: 32nMAssay Description:Inhibition of BRD3-BD1/2 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617014(CHEMBL5434556)
Affinity DataIC50: 35nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617032(CHEMBL5412288)
Affinity DataIC50: 37nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 38nMAssay Description:Inhibition of BRD3-BD1/2 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617033(CHEMBL5422341)
Affinity DataIC50: 46nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617018(CHEMBL5405976)
Affinity DataIC50: 63nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 78nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617025(CHEMBL5439531)
Affinity DataIC50: 80nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617012(CHEMBL5418334)
Affinity DataIC50: 83nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617026(CHEMBL5403237)
Affinity DataIC50: 100nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617029(CHEMBL5394293)
Affinity DataIC50: 100nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617019(CHEMBL5402033)
Affinity DataIC50: 100nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617031(CHEMBL5397542)
Affinity DataIC50: 100nMAssay Description:Inhibition of EZH2 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase EZH1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617034(CHEMBL5419363)
Affinity DataIC50: 124nMAssay Description:Inhibition of EZH1 (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617014(CHEMBL5434556)
Affinity DataIC50: 147nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617016(CHEMBL5432825)
Affinity DataIC50: 154nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617015(CHEMBL5434041)
Affinity DataIC50: 173nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617018(CHEMBL5405976)
Affinity DataIC50: 187nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617013(CHEMBL5427802)
Affinity DataIC50: 214nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617017(CHEMBL5431304)
Affinity DataIC50: 278nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617032(CHEMBL5412288)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617019(CHEMBL5402033)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617012(CHEMBL5418334)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617020(CHEMBL5395872)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617021(CHEMBL5408520)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617033(CHEMBL5422341)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617022(CHEMBL5426154)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617031(CHEMBL5397542)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617030(CHEMBL5393990)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617029(CHEMBL5394293)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617028(CHEMBL5417707)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617027(CHEMBL5436066)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50617026(CHEMBL5403237)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 (unknown origin) by HTRF analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
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