Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50019233
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616987(CHEMBL5400785)
Affinity DataIC50: 120nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616994(CHEMBL5401343)
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616981(CHEMBL5436028)
Affinity DataIC50: 263nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616988(CHEMBL5432118)
Affinity DataIC50: 385nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616989(CHEMBL5439633)
Affinity DataIC50: 437nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616992(CHEMBL5407344)
Affinity DataIC50: 443nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616980(CHEMBL5417528)
Affinity DataIC50: 835nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616977(CHEMBL5404938)
Affinity DataIC50: 960nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616990(CHEMBL5416613)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616986(CHEMBL5420819)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616983(CHEMBL5396275)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616982(CHEMBL5399237)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616978(CHEMBL5397867)
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616985(CHEMBL5401948)
Affinity DataIC50: 2.57E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616979(CHEMBL5403215)
Affinity DataIC50: 2.79E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616984(CHEMBL5394610)
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616991(CHEMBL5421771)
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616995(CHEMBL5435535)
Affinity DataIC50: 4.35E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616993(CHEMBL5422167)
Affinity DataIC50: 6.78E+3nMAssay Description:Inhibition of N-terminal His tagged recombinant human PTP1B expressed in Escherichia coli using pNPP as substrate assessed as substrate hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616987(CHEMBL5400785)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of recombinant human TC-PTP (1 to 314 residues) expressed in baculovirus infected insect cells using pNPP as substrate assessed as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616981(CHEMBL5436028)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human TC-PTP (1 to 314 residues) expressed in baculovirus infected insect cells using pNPP as substrate assessed as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616988(CHEMBL5432118)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human TC-PTP (1 to 314 residues) expressed in baculovirus infected insect cells using pNPP as substrate assessed as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616992(CHEMBL5407344)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human TC-PTP (1 to 314 residues) expressed in baculovirus infected insect cells using pNPP as substrate assessed as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Human)
Qingdao University

Curated by ChEMBL
LigandPNGBDBM50616994(CHEMBL5401343)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human TC-PTP (1 to 314 residues) expressed in baculovirus infected insect cells using pNPP as substrate assessed as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed