Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50019230
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616961(CHEMBL5419556)
Affinity DataKd:  160nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616962(CHEMBL5419190)
Affinity DataKd:  83nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616963(CHEMBL5403662)
Affinity DataKd:  78nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616964(CHEMBL5432442)
Affinity DataKd:  70nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616965(CHEMBL5398941)
Affinity DataKd:  92nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616966(CHEMBL5403329)
Affinity DataKd:  230nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616967(CHEMBL5433218)
Affinity DataKd:  150nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616968(CHEMBL5440251)
Affinity DataKd:  9.70nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50616969(CHEMBL5423528)
Affinity DataKd:  40nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50233225(CHEMBL4071864 | US12065447, Compound GSK2982772)
Affinity DataKd:  49nMAssay Description:Binding affinity to recombinant RIPK1 (unknown origin) assessed as dissociation constant by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed