Compile Data Set for Download or QSAR
Report error Found 113 Enz. Inhib. hit(s) with all data for entry = 50019224
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616870(CHEMBL5431371)
Affinity DataKi:  10nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616864(CHEMBL5412229)
Affinity DataKi:  12nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616861(CHEMBL5397812)
Affinity DataKi:  13nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616863(CHEMBL5410957)
Affinity DataKi:  13nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616868(CHEMBL5408011)
Affinity DataKi:  14nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616858(CHEMBL5425008)
Affinity DataKi:  16nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616869(CHEMBL5406204)
Affinity DataKi:  18nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616866(CHEMBL5408432)
Affinity DataKi:  20nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616856(CHEMBL5439290)
Affinity DataKi:  22nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616871(CHEMBL5403056)
Affinity DataKi:  27nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616875(CHEMBL5437241)
Affinity DataKi:  27nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616879(CHEMBL5427872)
Affinity DataKi:  28nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616892(CHEMBL5434126)
Affinity DataKi:  32nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616876(CHEMBL5404573)
Affinity DataKi:  36nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616893(CHEMBL5439899)
Affinity DataKi:  38nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616862(CHEMBL5404085)
Affinity DataKi:  40nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616859(CHEMBL5402597)
Affinity DataKi:  42nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616857(CHEMBL5419799)
Affinity DataKi:  44nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616871(CHEMBL5403056)
Affinity DataKi:  46nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616867(CHEMBL5395401)
Affinity DataKi:  47nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616865(CHEMBL5413838)
Affinity DataKi:  51nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616890(CHEMBL5426774)
Affinity DataKi:  52nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616866(CHEMBL5408432)
Affinity DataKi:  59nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616891(CHEMBL5402112)
Affinity DataKi:  65nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616861(CHEMBL5397812)
Affinity DataKi:  67nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616876(CHEMBL5404573)
Affinity DataKi:  67nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616877(CHEMBL5437741)
Affinity DataKi:  70nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616875(CHEMBL5437241)
Affinity DataKi:  71nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616888(CHEMBL5396978)
Affinity DataKi:  71nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616878(CHEMBL5409819)
Affinity DataKi:  79nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616864(CHEMBL5412229)
Affinity DataKi:  83nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616860(CHEMBL5435516)
Affinity DataKi:  85nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616868(CHEMBL5408011)
Affinity DataKi:  95nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616870(CHEMBL5431371)
Affinity DataKi:  99nMAssay Description:Binding affinity to 5-HT1D receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616881(CHEMBL5397921)
Affinity DataKi:  105nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616874(CHEMBL5406365)
Affinity DataKi:  108nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616881(CHEMBL5397921)
Affinity DataKi:  110nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616882(CHEMBL5419212)
Affinity DataKi:  112nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616879(CHEMBL5427872)
Affinity DataKi:  122nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616886(CHEMBL5416938)
Affinity DataKi:  129nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616877(CHEMBL5437741)
Affinity DataKi:  132nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616889(CHEMBL5423305)
Affinity DataKi:  134nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616863(CHEMBL5410957)
Affinity DataKi:  137nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616865(CHEMBL5413838)
Affinity DataKi:  155nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616872(CHEMBL5421590)
Affinity DataKi:  155nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616888(CHEMBL5396978)
Affinity DataKi:  159nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616892(CHEMBL5434126)
Affinity DataKi:  159nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616870(CHEMBL5431371)
Affinity DataKi:  165nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616883(CHEMBL5403411)
Affinity DataKi:  165nMAssay Description:Displacement of [3H](+)-ditolylguanidine from human sigma 2 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligan...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50616886(CHEMBL5416938)
Affinity DataKi:  166nMAssay Description:Displacement of [3H](+)-pentazocine from human sigma 1 receptor transfected in human HEK293T cells assessed as inhibition constant by radioligand com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
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