Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50018183
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405853(CHEMBL5273189)
Affinity DataEC50:  900nMAssay Description:Inverse agonist activity at human GPR55 expressed in HEK293 cells coexpressing serum response element assessed as reduction in MAPK/ERK signalling pa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405853(CHEMBL5273189)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM61535([4-(2,7-dimethyl-5,6,7,8-tetrahydro-[1]benzothiolo...)
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human GPR55 expressed in human U2OS cells assessed as inhibition of LPI-induced receptor activation by measuring beta-arrestin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM61528(cid_1261290 | N-(4-{[(3,4-dimethyl-5-isoxazolyl)am...)
Affinity DataIC50: 500nMAssay Description:Antagonist activity at GPR55 (unknown origin) by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405850(CHEMBL5273001)
Affinity DataIC50: 680nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM61427(SMR000116779 | furan-2-yl-[4-(2-methyl-5,6,7,8-tet...)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at GPR55 (unknown origin) by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM61399(SMR000003886 | [4-(2-cyclopropyl-5,6,7,8-tetrahydr...)
Affinity DataIC50: 860nMAssay Description:Antagonist activity at human GPR55 expressed in human U2OS cells assessed as inhibition of LPI-induced receptor activation by measuring beta-arrestin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405870(CHEMBL5275934)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at GPR55 (unknown origin) by beta-arrestin recruitment assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405853(CHEMBL5273189)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human GPR55 expressed in HEK293 cells coexpressing serum response element assessed as inhibition of LPI-induced MAPK/ERK signa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM61427(SMR000116779 | furan-2-yl-[4-(2-methyl-5,6,7,8-tet...)
Affinity DataIC50: 2.02E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405861(CHEMBL5278819)
Affinity DataIC50: 2.14E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405852(CHEMBL5281110)
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405854(CHEMBL5282587)
Affinity DataIC50: 2.78E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405859(CHEMBL5271818)
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405858(CHEMBL5275607)
Affinity DataIC50: 3.35E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405855(CHEMBL5267293)
Affinity DataIC50: 7.16E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM61427(SMR000116779 | furan-2-yl-[4-(2-methyl-5,6,7,8-tet...)
Affinity DataIC50: 7.50E+3nMAssay Description:Antagonist activity at human GPR55 expressed in HEK293 cells coexpressing serum response element assessed as inhibition of LPI-induced MAPK/ERK signa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405860(CHEMBL5278170)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405851(CHEMBL5283686)
Affinity DataIC50: 9.49E+3nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405856(CHEMBL5267388)
Affinity DataIC50: 1.17E+4nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405857(CHEMBL5281025)
Affinity DataIC50: 2.93E+4nMAssay Description:Antagonist activity at beta-galactosidase fused human GPR55 expressed in CHO cells assessed as inhibition of LPI-induced receptor activation by measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405866(CHEMBL5267725)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405865(CHEMBL5286922)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405850(CHEMBL5273001)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405851(CHEMBL5283686)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405853(CHEMBL5273189)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405854(CHEMBL5282587)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405867(CHEMBL5283527)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405868(CHEMBL5285121)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405869(CHEMBL5289588)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405855(CHEMBL5267293)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405859(CHEMBL5271818)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405860(CHEMBL5278170)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405862(CHEMBL5270755)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405868(CHEMBL5285121)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405864(CHEMBL5285314)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405865(CHEMBL5286922)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405866(CHEMBL5267725)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405850(CHEMBL5273001)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405851(CHEMBL5283686)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405853(CHEMBL5273189)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405854(CHEMBL5282587)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405867(CHEMBL5283527)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405863(CHEMBL5284821)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405869(CHEMBL5289588)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405855(CHEMBL5267293)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405859(CHEMBL5271818)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405860(CHEMBL5278170)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405862(CHEMBL5270755)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405863(CHEMBL5284821)
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition constant incubated for 90 mins by liqui...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
Displayed 1 to 50 (of 51 total ) | Next | Last >>
Jump to: