Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50019512
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620061(CHEMBL5401025)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620062(CHEMBL5414217)
Affinity DataIC50: 2nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620069(CHEMBL5426778)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620060(CHEMBL5398050)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620070(CHEMBL5418588)
Affinity DataIC50: 15nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620071(CHEMBL5404185)
Affinity DataIC50: 22nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620068(CHEMBL5403184)
Affinity DataIC50: 26nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620063(CHEMBL5412890)
Affinity DataIC50: 33nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620064(CHEMBL5427001)
Affinity DataIC50: 47nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620066(CHEMBL5394271)
Affinity DataIC50: 69nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620067(CHEMBL5430269)
Affinity DataIC50: 75nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50620065(CHEMBL5432829)
Affinity DataIC50: 140nMAssay Description:Inhibition of TNKS1 (unknown origin) using biotinylated NAD as substrate preincubated for 30 mins followed by substrate addition and measured after 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed