Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50019331
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  14nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataKd:  686nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  9nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataKd:  419nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  9nMAssay Description:Binding affinity to BRD2 BD2 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataKd:  1.75E+4nMAssay Description:Binding affinity to BRD2 BD2 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  11nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataKd:  7.43E+3nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) by thermal denaturation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 0.820nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618177(CHEMBL5408527)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618176(CHEMBL5396203)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618175(CHEMBL5406617)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618172(CHEMBL5416735)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618179(CHEMBL5405309)
Affinity DataIC50: 2nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618173(CHEMBL5394959)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618178(CHEMBL5423358)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618180(CHEMBL5435358)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 17nMAssay Description:Inhibition of BRD2 bromodomain 2 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 22nMAssay Description:Inhibition of BRD4 bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 39nMAssay Description:Inhibition of BRD3 bromodomain 2 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 64nMAssay Description:Inhibition of BRD3 bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 69nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 134nMAssay Description:Inhibition of BRDT bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 155nMAssay Description:Inhibition of BRD2 bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 820nMAssay Description:Inhibition of BRD4 bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of BRD4 bromodomain 2 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of BRD2 bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of BRD3 bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of BRDT bromodomain 1 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of BRD2 bromodomain 2 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50618174(CHEMBL5427713)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of BRD3 bromodomain 2 (unknown origin) by Alphascreen based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed