Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50020736
TargetFibroblast growth factor receptor 1(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 34nMAssay Description:Inhibition of FGFR-1 (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant EGFR (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633199(CHEMBL5398753)
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 1(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633199(CHEMBL5398753)
Affinity DataIC50: 82nMAssay Description:Inhibition of FGFR-1 (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50595124(VANDETANIB | CHEBI:49960 | Vandetanib | GNF-PF-218...)
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633199(CHEMBL5398753)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant EGFR (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633204(CHEMBL5395205)
Affinity DataIC50: 108nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633202(CHEMBL5404512)
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633200(CHEMBL5415189)
Affinity DataIC50: 242nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633203(CHEMBL5402749)
Affinity DataIC50: 438nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633205(CHEMBL5396585)
Affinity DataIC50: 455nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandPNGBDBM50633201(CHEMBL5399404)
Affinity DataIC50: 536nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed