Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50020730
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50221516(6-methoxy-7-(3-morpholinopropoxy)-4-((1R,2S)-2-phe...)
Affinity DataIC50: 5nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM4445(4-[(3-bromophenyl)amino]-6,7-dimethoxyquinoline-3-...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)
Affinity DataIC50: 110nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) using poly (Glu,Tyr) as substrate incubated for 40 mins in presence of ATP by Kinase-Glo lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50633121(CHEMBL5410384)
Affinity DataIC50: 138nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) using poly (Glu,Tyr) as substrate incubated for 40 mins in presence of ATP by Kinase-Glo lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50633120(CHEMBL5404784)
Affinity DataIC50: 144nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) using poly (Glu,Tyr) as substrate incubated for 40 mins in presence of ATP by Kinase-Glo lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50633118(CHEMBL5408255)
Affinity DataIC50: 152nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) using poly (Glu,Tyr) as substrate incubated for 40 mins in presence of ATP by Kinase-Glo lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50633119(CHEMBL5438940)
Affinity DataIC50: 159nMAssay Description:Inhibition of EGFR L858R/T790M mutant (unknown origin) using poly (Glu,Tyr) as substrate incubated for 40 mins in presence of ATP by Kinase-Glo lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50633122(CHEMBL5416668)
Affinity DataIC50: 490nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50517778(CHEMBL4447196)
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50117655(CHEMBL3613691)
Affinity DataIC50: 5.28E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM50599337(CHEMBL5206476)
Affinity DataIC50: 5.30E+6nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Radhabai Kale Mahila Mahavidyalaya

Curated by ChEMBL
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataIC50: 8.30E+7nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed