Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50016576
TargetProtein-arginine deiminase type-4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50595779(CHEMBL5180282)
Affinity DataIC50: 14nMAssay Description:Inhibition of human His-Sumo-tagged PAD4 (A2 to P663 residues) expressed in Escherichia coli BL21 (DE3) cells using BAEE as substrate preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein-arginine deiminase type-4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50595777(CHEMBL5187676)
Affinity DataIC50: 17nMAssay Description:Inhibition of human His-Sumo-tagged PAD4 (A2 to P663 residues) expressed in Escherichia coli BL21 (DE3) cells using BAEE as substrate preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein-arginine deiminase type-4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50595776(CHEMBL5201255)
Affinity DataIC50: 19nMAssay Description:Inhibition of human His-Sumo-tagged PAD4 (A2 to P663 residues) expressed in Escherichia coli BL21 (DE3) cells using BAEE as substrate preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein-arginine deiminase type-4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50595775(CHEMBL5188806)
Affinity DataIC50: 20nMAssay Description:Inhibition of human His-Sumo-tagged PAD4 (A2 to P663 residues) expressed in Escherichia coli BL21 (DE3) cells using BAEE as substrate preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein-arginine deiminase type-4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50595778(CHEMBL5195279)
Affinity DataIC50: 20nMAssay Description:Inhibition of human His-Sumo-tagged PAD4 (A2 to P663 residues) expressed in Escherichia coli BL21 (DE3) cells using BAEE as substrate preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein-arginine deiminase type-4(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50595780(CHEMBL5194669)
Affinity DataIC50: 22nMAssay Description:Inhibition of human His-Sumo-tagged PAD4 (A2 to P663 residues) expressed in Escherichia coli BL21 (DE3) cells using BAEE as substrate preincubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed