Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50016562
TargetTyrosine-protein kinase JAK3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595733(CHEMBL5192697)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of JAK3 (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595734(CHEMBL5197209)
Affinity DataIC50: 9nMAssay Description:Inhibition of JAK3 (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595732(CHEMBL5202699)
Affinity DataIC50: 16nMAssay Description:Inhibition of BTK (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595735(CHEMBL5178256)
Affinity DataIC50: 33nMAssay Description:Inhibition of JAK3 (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595733(CHEMBL5192697)
Affinity DataIC50: 98nMAssay Description:Inhibition of BTK (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595735(CHEMBL5178256)
Affinity DataIC50: 638nMAssay Description:Inhibition of BTK (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595732(CHEMBL5202699)
Affinity DataIC50: 699nMAssay Description:Inhibition of JAK3 (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595736(CHEMBL5207244)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-AEPF-pNA peptide as substrate incubated for 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetTyrosine-protein kinase BTK(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595734(CHEMBL5197209)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BTK (unknown origin) using TK peptide as substrate incubated for 1 hr in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50595737(CHEMBL5206882)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of GST-tagged Pin1 (unknown origin) using Suc-AEPF-pNA peptide as substrate incubated for 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed