Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50035696
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024594(LEUCINE PHOSPHONIC ACID | (R)-1-Ammonium-3-methyl-...)
Affinity DataKi:  230nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024596([(1R)-1-amino-2-phenylethyl]phosphonic acid | (R)-...)
Affinity DataKi:  420nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024590(1-Ammonium-octane-1-phosphonic acid anion | CHEMBL...)
Affinity DataKi:  470nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024601(1-aminohexylphosphonic acid | 1-Ammonium-hexane-1-...)
Affinity DataKi:  1.00E+3nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024602(1-amino-2-methylpropylphosphonic acid | 1-Ammonium...)
Affinity DataKi:  1.20E+3nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024604(1-aminopropylphosphonic acid | 1-Ammonium-propane-...)
Affinity DataKi:  3.60E+3nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024592((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...)
Affinity DataKi:  1.54E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024608(1-[amino({[(1S)-1-carboxylate anion-3-methylbutyl]...)
Affinity DataKi:  4.00E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024599((1-Ammonium-2-phenyl-ethyl)-phosphonic acid monome...)
Affinity DataKi:  4.30E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024588(2-{[(1-Ammonium-3-methyl-butyl)-hydroxy-phosphinoy...)
Affinity DataKi:  5.60E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024598(2-[(1-Ammonium-3-methyl-butyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  5.80E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50078139((1-Ammonium-2-phenyl-ethyl)-phosphinic acid | (1-A...)
Affinity DataKi:  5.90E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50078132((1-Amino-3-methyl-butyl)-phosphinic acid | (1-Ammo...)
Affinity DataKi:  8.70E+4nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024597((S)-1-Ammonium-3-methyl-butane-1-phosphonic acid a...)
Affinity DataKi:  2.20E+5nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50017377(1-Ammonium-ethanephosphonic acid anion | 1-aminoet...)
Affinity DataKi:  2.40E+5nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024606((1-Ammonium-3-methyl-butyl)-phosphonic acid monome...)
Affinity DataKi:  3.20E+5nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024607(2-[(1-Ammonium-2-phenyl-ethyl)-hydroxy-phosphinoyl...)
Affinity DataKi:  3.40E+5nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024593((3-Methyl-butyl)-phosphonic acid | CHEMBL41600)
Affinity DataKi:  7.75E+5nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024600(2-(1-Ammonium-3-methylbutylmethoxyphosphorylcarbon...)
Affinity DataKi:  1.65E+6nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024591(Ammonium-methanephosphonic acid anion | CHEMBL4187...)
Affinity DataKi:  1.04E+6nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50024589(3-Methyl-butylamine | 3-METHYLBUTAN-1-AMINE | CHEM...)
Affinity DataKi: >5.00E+7nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed