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Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50018056
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607268(CHEMBL5220657)
Affinity DataIC50: 0.130nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607267(CHEMBL5220613)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607263(CHEMBL5220594)
Affinity DataIC50: 0.160nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607273(CHEMBL5219939)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607269(CHEMBL5220750)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607275(CHEMBL5219299)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607276(CHEMBL5219451)
Affinity DataIC50: 0.280nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607265(CHEMBL5219532)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50228403(8-[(3R)-3-Aminopiperidin-1-yl]-7-but-2-yn-1-yl-3-m...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate incubated for 30 mins by continuous fluorescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607278(CHEMBL5220474)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607271(CHEMBL5218500)
Affinity DataIC50: 0.75nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607277(CHEMBL5219735)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50225074(CHEMBL385517 | BMS-477118 | (1S,6S)-2-(2-adamantan...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate incubated for 30 mins by continuous fluorescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607274(CHEMBL5220415)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607266(CHEMBL5219761)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate incubated for 30 mins by continuous fluorescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607279(CHEMBL5219966)
Affinity DataIC50: 10nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607270(CHEMBL5220348)
Affinity DataIC50: 15nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM126822(US8785477, Sitagliptin)
Affinity DataIC50: 18nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate incubated for 30 mins by continuous fluorescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM126822(US8785477, Sitagliptin)
Affinity DataIC50: 19nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607272(CHEMBL5220053)
Affinity DataIC50: 25nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate incubated for 30 mins by continuous fluorescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Guru Nanak Dev University

Curated by ChEMBL
LigandPNGBDBM50607264(CHEMBL5219996)
Affinity DataIC50: 171nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by fluorescence based enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed